Product Name |
Dendrotoxin K TFA |
Cat. No. |
TD-HYP3089A |
Description |
Dendrotoxin K TFA 是一种 Kv1.1 通道阻滞剂。Dendrotoxin K TFA 通过控制突触前尖峰波以时间依赖性方式将谷氨酸释放入 CA3 神经元中。 |
Purity |
99.54% |
分子式 |
C₂₉₄H₄₆₂N₈₄O₇₅S₆・XC₂HF₃OC₂ |
分子量 |
6559.66 (free base) |
Sequence |
Ala-Ala-Lys-Tyr-Cys-Lys-Leu-Pro-Leu-Arg-Ile-Gly-Pro-Cys-Lys-Arg-Lys-Ile-Pro-Ser-Phe-Tyr-Tyr-Lys-Trp-Lys-Ala-Lys-Gln-Cys-Leu-Pro-Phe-Asp-Tyr-Ser-Gly-Cys-Gly-Gly-Asn-Ala-Asn-Arg-Phe-Lys-Thr-Ile-Glu-Glu-Cys-Arg-Arg-Thr-Cys-Val-Gly (Disulfide bridge:Cys5-Cys55,Cys14-Cys38,Cys30-Cys51) |
Sequence Shortening |
AAKYCKLPLRIGPCKRKIPSFYYKWKAKQCLPFDYSGCGGNANRFKTIEECRRTCVG (Disulfide bridge:Cys5-Cys55,Cys14-Cys38,Cys30-Cys51) |
作用靶点 |
Potassium Channel |
作用通路 |
Membrane Transporter/Ion Channel |
储存方式 |
Sealed storage, away from moisture and light, under nitrogen
Powder: -80°C, 2 years;-20°C, 1 year
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light, under nitrogen) |