c(RGD)环肽:c(RGDfV)、c(RGD-DPhe-V)
描 述:Cyclo(Arg-Gly-Asp-D-Phe-Val) (Cyclo(RGDfV)) 是一种整合素 αvβ3 抑制剂。Cyclo(Arg-Gly-Asp-D-Phe-Val) 具有抗肿瘤活性。Cyclo(Arg-Gly-Asp-D-Phe-Val) 可用于急性髓系白血病的研究。
CAS号:137813-35-5
单字母: Cyclo(RGDfV)
多字母:Cyclo(Arg-Gly-Asp-DPhe-Val)
分子式: C26H38N8O7
分子量: 574.63
参考文献:[1]. Shen ZH, et al. Targeting of the leukemia microenvironment by c(RGDfV) overcomes the resistance to chemotherapy in acute myeloid leukemia in biomimetic polystyrene scaffolds. Oncol Lett. 2016 Nov;12(5):3278-3284.